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Synthesis and fungicidal activities of a novel series of 4-[3-(Pyrid-4-yl)-3-substituted phenyl acryloyl] morpholine

文献类型： 外文期刊

作者： Mu Chang-Wei 1 ; Yuan Hui-Zhu 1 ; Li Nan 1 ; Fu Bin 1 ; Xiao Yu-Mei 1 ; Ma Yong-Qiang 1 ; Qi Shu-Hua 1 ; Qin Zhao-Hai 1 ;

作者机构： 1.China Agr Univ, Coll Sci, Beijing 100094, Peoples R China; Chinese Acad Agr Sci, Inst Plant Protect, Beijing 100094, Peoples R China

关键词： pyridine derivative;acryloyl morpholine;fungicidal activity

期刊名称：CHEMICAL JOURNAL OF CHINESE UNIVERSITIES-CHINESE （ 影响因子：0.65； 五年影响因子：0.481 ）

ISSN： 0251-0790

年卷期： 2007 年 28 卷 10 期

页码：

收录情况： SCI

摘要： In searching for novel and high active fungicides with pyridyl moiety, with Dimethomorph as a model compound and isonicotinic acid as the main starting material, twenty-seven title compounds were designed and synthesized through chlorination, Friedel-Crafts acylation, Wittig-Horner reaction and other steps. All the target structures were confirmed via H-1 NMR and elementary analysis. In the preliminary fungicidal evaluation, all the compounds exhibit a significant inhibiting activity against Rhizoctonia solanti Kuhn and Phytophthora drechsler Tucker. Among them, the EC50 values of compounds 4-20, 4-21 and 4-22 to Rhizoctonia solani Kuhn were 28. 94, 5. 27 and 0. 87 mu g/mL, respectively, compared to 1. 54 mu g/mL of Carbendazim and 60. 95 mu g/mL of Dimethomorph; and to Phytophthora drechsler Tucker were 0. 33, 0. 27 and 0. 09 mu/mL, respectively, compared to 20. 39 mu/mL of Chlorothalonil and 0. 24 mu g/mL of Dimethomorph. The results suggest that they might be valuable in the control of plant diseases.

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